Increase serotonin release
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Amphetamines, MDMA
Antidepressants: mirtazapine
Opioids: oxycodone, tramadol, dextromethorphan
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Inhibit serotonin uptake
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Amphetamines, MDMA, cocaine
SSRIs: citalopram, escitalopram, fluoxetine, paroxetine, sertraline
SNRIs: duloxetine, venlafaxine
TCAs: amitriptyline, clomipramine, imipramine
Opioids: methadone, tramadol, dextromethorphan
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Inhibit serotonin metabolism
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Anxiolytics: buspirone
MAOI: phenelzine, rasagiline, selegiline
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Activate Serotonin Receptors
Inhibit Cytochrome P450
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Hallucinogen: LSD
Antidepressants: trazodone
Opioids: fentanyl
Mood stabilizers: lithium
CYP2D6
Inhibitors: fluoxetine, sertraline
Substrates: dextromethorphan, oxycodone, risperidone, tramadol
CYP3A4
Inhibitors: ciprofloxacin, ritonavir
Substrates: methadone, oxycodone, venlafaxine
CYP2C19
Inhibitors: fluconazole
Substrates: citalopram
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